Metabolic Compound

Orforglipron

First oral non-peptide GLP-1 receptor agonist (Eli Lilly); Phase 3 obesity program.

Scientific Overview

Orforglipron (LY3502970) is Eli Lilly's small-molecule, non-peptide GLP-1R agonist. Unlike oral semaglutide it does not require SNAC absorption enhancers or fasted dosing. Phase 2 obesity (2023) showed up to 14.7% weight loss at 36 weeks. Phase 3 ATTAIN and ACHIEVE programs read out in 2025.

Key Research Benefits

  • Oral once-daily dosing
  • No food/water restrictions
  • Weight loss comparable to injectable GLP-1s in Phase 2

Potential Side Effects

Nausea
Vomiting
Diarrhea
Constipation

Research Protocols

Common Dosages

Investigational

12 -> 36 mg
Daily, oral

Phase 3 dose range

Note: Dosages listed are common research protocols found in peer-reviewed literature and clinical trials. Individual results and requirements may vary significantly in a research context.

Dose Calculator

🧮 Peptide Reconstitution Calculator

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480 Units

or 4.80 mL on a U-100 syringe

Concentration:2.50 mg/mL
Peptide per Unit:25.00 mcg/unit
*Always double-check your calculations. This tool is for educational purposes only.

Explore Orforglipron

Orforglipron by goal

Read Orforglipron's profile filtered through specific research goals.

Molecular Profile

small-molecule
C44H52FN7O5
1 AA Sequence

Quick Reference

Status
Research Compound
Category
Metabolic
Common Dosage
12 -> 36 mg
Daily, oral

Strictly for research purposes. Not for human consumption.

Medical Disclaimer

Information provided on DoseVault is for educational and research purposes only. This website does not advocate for the human use of peptides. Peptides are currently sold as research chemicals and are not FDA-approved for human consumption. Always consult a licensed medical professional before considering any protocol.